Consumer medicine information

Celecoxib BTC Capsules

Celecoxib

BRAND INFORMATION

Brand name

Celecoxib BTC

Active ingredient

Celecoxib

Schedule

S4

 

Consumer medicine information (CMI) leaflet

Please read this leaflet carefully before you start using Celecoxib BTC Capsules.

What is in this leaflet

Read this leaflet carefully before taking your medicine.

This leaflet answers some common questions about celecoxib. It does not contain all the available information. It does not take the place of talking to your doctor or pharmacist.

The information in this leaflet was last updated on the date listed on the last page. More recent information on this medicine may be available.

Ask your doctor or pharmacist:

  • if there is anything you do not understand in this leaflet,
  • if you are worried about taking your medicine, or
  • to obtain the most up-to-date information.

You can also download the most up to date leaflet from www.apotex.com.au.

All medicines have risks and benefits. Your doctor has weighed the risks of you using this medicine against the benefits they expect it will have for you.

Pharmaceutical companies cannot give you medical advice or an individual diagnosis.

Keep this leaflet with your medicine. You may want to read it again.

What this medicine is used for

The name of your medicine is Celecoxib BTC. It contains the active ingredient celecoxib.

It is used to treat:

  • osteoarthritis,
  • rheumatoid arthritis
  • ankylosing spondylitis, a chronic inflammatory rheumatic disorder that primarily affects, but is not limited to, the spine.

Celecoxib also provides short term pain relief in conditions such as:

  • menstrual cramps or period pain
  • after surgery
  • muscle and joint injuries.

Ask your doctor if you have any questions about why this medicine has been prescribed for you. Your doctor may have prescribed this medicine for another reason.

This medicine is available only with a doctor's prescription.

How it works

Celecoxib belongs to a group of medicines called Coxibs which are used to relieve pain and inflammation in a number of conditions. Although Celecoxib BTC can relieve the symptoms of pain and inflammation, it will not cure your condition.

There is no evidence that this medicine is addictive.

Use in children

This medicine should not be used in children or adolescents under 18 years of age.

Before you take this medicine

When you must not take it

Do not take this medicine if:

  • You have or have had any of the following:
    - severe heart disease
    - blood vessel disease affecting the circulation in your brain or limbs
    - severe liver problems
    - recently undergone a coronary artery bypass graft
    - peptic ulceration or gastric intestinal bleeding
    - severe kidney problems
    - an attack of asthma, hives, itching, skin rash or a runny nose after taking Aspirin or other Non-Steroidal Anti-Inflammatory Drugs (NSAIDs), including other Coxib medicines.
  • You are taking any other NSAIDs.
  • You are hypersensitive to, or have had an allergic reaction to, celecoxib, any of the ingredients listed at the end of this leaflet or sulfonamides, a group of medicines which include certain antibiotics (if you are not sure if you are taking one of these medicines ask your doctor or pharmacist).
    Symptoms of an allergic reaction may include: shortness of breath, wheezing or difficulty breathing; swelling of the face, lips, tongue, throat or other parts of the body; rash, itching or hives on the skin; fainting; or hay fever-like symptoms.
    If you think you are having an allergic reaction, do not take any more of the medicine and contact your doctor immediately or go to the Accident and Emergency department at the nearest hospital.
  • The expiry date (EXP) printed on the pack has passed.
  • The packaging is torn, shows signs of tampering or it does not look quite right.

Before you start to take it

Before you start taking this medicine, tell your doctor if:

  1. You have allergies to:
  • any other medicines
  • any other substances, such as foods, preservatives or dyes.
  1. You have or have had any medical conditions, especially the following:
  • diabetes
  • high blood pressure or fluid retention
  • high cholesterol levels
  • heart failure
  • history of heart problems or stroke
  • circulation problems in your limbs
  • liver or kidney problems
  • asthma, hives, itching, skin rash or runny nose
  • peptic ulcer
  • vomiting blood or material that looks like coffee grounds
  • bleeding from the rectum, have black sticky bowel motions or bloody diarrhoea
  • low blood count
  • inflammatory bowel disease
  • infection.
  1. You are currently pregnant or you plan to become pregnant. Do not take this medicine whilst pregnant until you and your doctor have discussed the risks and benefits involved.
  2. You are currently breastfeeding or you plan to breastfeed. Do not take this medicine whilst breastfeeding until you and your doctor have discussed the risks and benefits involved.
NSAIDs, which are related medicines, have been associated with reversible infertility in some women.
Use of NSAIDS in early pregnancy can increase the risk of spontaneous abortion.
There is no information on the use of Celecoxib BTC during pregnancy.
Celecoxib BTC may affect your developing baby if taken during pregnancy. Particular caution should be exerted from the twentieth week of pregnancy.
  1. You drink large amounts of alcohol.
  2. You are a smoker.
  3. You are currently receiving or are planning to receive dental treatment.
  4. You are planning to have surgery.
  5. You are taking or are planning to take any other medicines. This includes vitamins and supplements that are available from your pharmacy, supermarket or health food shop.

Some medicines may interact with celecoxib. These include:

  • medicines to treat high blood pressure and some other heart problems such as ACE inhibitors, angiotensin receptor antagonists, beta-blockers and diuretics (also called fluid or water tablets)
  • frusemide and thalizides, types of diuretics
  • aspirin
  • metoprolol, a beta-blocker used for heart conditions, high blood pressure and migraines
  • fluconazole, an antifungal agent
  • lithium, a medicine used to treat some types of mood disorders
  • warfarin, apixaban, dabigatran, and rivaroxaban, medicines used to stop blood clots
  • rifampicin, an antibiotic
  • carbamazepine, a medicine used for epilepsy
  • barbiturates, a class of medicines that cause sedation
  • cyclosporin, an immune suppressant
  • antacids, medicines used to treat indigestion
  • dextromethorphan, a cough suppressant
  • medicines used to treat pain and inflammation called Non-Steroidal Anti-Inflammatory Drugs (NSAIDs) or (cortico) steroids.

If you are taking any of these you may need a different dose or you may need to take different medicines.

Other medicines not listed above may also interact with celecoxib.

How to take this medicine

Follow carefully all directions given to you by your doctor. Their instructions may be different to the information in this leaflet.

How much to take

Your doctor will tell you how much of this medicine you should take. This will depend on your condition and whether you are taking any other medicines.

Do not stop taking your medicine or change your dosage without first checking with your doctor.

Osteoarthritis
The recommended dose is 200 mg once daily or 100 mg twice daily.

Rheumatoid arthritis
The recommended dose is 100 mg twice daily.

Ankylosing spondylitis
The maximum recommended dose is 200 mg once daily or 100 mg twice daily.

Menstrual cramps or period pain
The recommended dose is 400 mg as a single dose on the first day and 200 mg once daily on the following days. The maximum recommended treatment duration is 5 days.

Muscle and joint injuries or after surgery
The recommended dose is 400 mg as a first dose followed by 200 mg once or twice daily as required for up to 5 days.

How to take it

Swallow the capsule whole with a glass of fluid.

When to take it

Take this medicine at the same time each day. Taking it at the same time each day will have the best effect and will also help you remember when to take it.

It does not matter if you take it before, with or after food.

How long to take it for

Continue taking your medicine for as long as your doctor tells you.

Make sure you have enough of this medicine to last over weekends and holidays.

If you forget to take it

If it is almost time to take your next dose, skip the missed dose and take your next dose at the usual time. Otherwise, take it as soon as you remember and then go back to taking your medicine as you would normally.

Do not take a double dose to make up for missed doses. This may increase the chance of you experiencing side effects.

If you have trouble remembering to take your medicine, ask your pharmacist for some hints to help you remember.

If you take too much (overdose)

If you think that you or anyone else may have taken too much of this medicine, immediately telephone your doctor or the Poisons Information Centre (Tel: 13 11 26 in Australia) for advice. Alternatively, go to the Accident and Emergency department at your nearest hospital.

Do this even if there are no signs of discomfort or poisoning. You may need urgent medical attention.

Signs of an overdose with celecoxib may include:

  • nausea and/or vomiting
  • headache
  • drowsiness/tiredness
  • difficulty in breathing
  • impaired consciousness
  • kidney failure.

While you are taking this medicine

Things you must do

Tell your doctor that you are taking this medicine if:

  • you are about to be started on any new medicine
  • you are pregnant or are planning to become pregnant
  • you are breastfeeding or are planning to breastfeed
  • you are about to have any blood tests
  • you are going to have surgery or are going into hospital.

Your doctor may occasionally do tests to make sure the medicine is working and to prevent side effects. Go to your doctor regularly for a check-up.

Tell any other doctors, dentists and pharmacists who are treating you that you take this medicine.

Things you must not do

Do not:

  • Give this medicine to anyone else, even if their symptoms seem similar to yours.
  • Take your medicine to treat any other condition unless your doctor tells you to.
  • Stop taking your medicine, or change the dosage, without first checking with your doctor.

Things to be careful of

Be careful when driving or operating machinery until you know how this medicine affects you.

Possible side effects

Tell your doctor or pharmacist as soon as possible if you do not feel well while you are taking celecoxib or if you have any questions or concerns.

Do not be alarmed by the following lists of side effects. You may not experience any of them. All medicines can have side effects. Sometimes they are serious but most of the time they are not.

Tell your doctor if you notice any of the following:

  • stomach pain, diarrhoea, indigestion, wind, nausea
  • back pain, swollen hands, ankles and feet, unexplained weight gain
  • dizziness
  • sore throat, runny nose, sinusitis, upper respiratory tract infection
  • skin rash
  • difficulty sleeping.

Tell your doctor as soon as possible if you notice any of the following.

These may be serious side effects and you may need medical attention:

  • blistering and bleeding in the lips, eyes, mouth, nose and genitals
  • swelling, blistering or peeling of the skin, which may be accompanied by fever, chills, headache, sore throat, diarrhoea, aching joints and muscles
  • severe stomach or throat pain, vomiting blood or black sticky bowel motions
  • bleeding or bruising more than usual, reddish or purple blotches under the skin
  • nausea, lethargy, itchiness, flulike symptoms or yellowing of the skin or eyes (jaundice)
  • signs of anaemia such as tiredness, being short of breath and looking pale
  • loss or deterioration of hearing
  • confusion
  • redness, irritation or watering of the eye(s)
  • experience sensations with any of the senses (sight, sound, touch, taste or feel) which may not be real
  • severe or persistent headache, fever, stiff neck, sensitivity to light and vomiting
  • worsening epilepsy.

Allergic reactions

If you think you are having an allergic reaction to celecoxib, do not take any more of this medicine and tell your doctor immediately or go to the Accident and Emergency department at your nearest hospital.

Symptoms of an allergic reaction may include some or all of the following:

  • , shortness of breath, wheezing or difficulty breathing
  • swelling of the face, lips, tongue, throat or other parts of the body
  • rash, itching or hives on the skin
  • fainting
  • hay fever-like symptoms.

Storage and disposal

Storage

Keep your medicine in its original packaging until it is time to take it.

If you take your medicine out of its original packaging it may not keep well.

Keep your medicine in a cool dry place where the temperature will stay below 25°C. Do not store your medicine, or any other medicine, in the bathroom or near a sink. Do not leave it on a window sill or in the car. Heat and dampness can destroy some medicines.

Keep this medicine where children cannot reach it. A locked cupboard at least one-and-a-half metres above the ground is a good place to store medicines.

Disposal

If your doctor tells you to stop taking this medicine or it has passed its expiry date, your pharmacist can dispose of the remaining medicine safely.

Product description

What Celecoxib BTC capsules look like

100 mg capsules: opaque, white to off-white capsules imprinted with 'CC' and '100' in black ink.

Blister pack of 60 capsules.

200 mg capsules: white to off-white capsules imprinted with 'CC' and '200' in black ink.

Blister pack of 30 capsules.

* Not all strengths may be available.

Ingredients

Each capsule contains 100 mg or 200 mg of celecoxib as the active ingredient.

It also contains the following inactive ingredients:

  • lactose monohydrate
  • povidone
  • colloidal anhydrous silica
  • sodium lauryl sulfate
  • croscarmellose sodium and
  • magnesium stearate

The capsule shell contains:

  • gelatin
  • titanium dioxide
  • sodium lauryl sulfate
  • TekPrint SW-9008 Black Ink (Proprietary Ingredient # 2328)

This medicine contains traces of sulfites. This medicine contains lactose. This medicine is gluten-free, sucrose-free, tartrazine-free and free of other azo dyes.

Australian Registration Numbers

Celecoxib BTC 100 mg capsules blister pack: AUST R 212786

Celecoxib BTC 200 mg capsules blister pack: AUST R 212788

Sponsor

Apotex Pty Ltd
16 Giffnock Avenue
Macquarie Park NSW 2113

This leaflet was last updated in December 2021.

Published by MIMS February 2022

BRAND INFORMATION

Brand name

Celecoxib BTC

Active ingredient

Celecoxib

Schedule

S4

 

1 Name of Medicine

Celecoxib.

2 Qualitative and Quantitative Composition

Each capsule contains 100 mg or 200 mg celecoxib as the active ingredient.
Excipients with known effect. Lactose monohydrate.
For the full list of excipients see Section 6.1 List of Excipients.

3 Pharmaceutical Form

Capsule, hard.
100 mg capsules: opaque, white to off-white capsules imprinted with 'CC' and '100' in black ink.
200 mg capsules: white to off-white capsules imprinted with 'CC' and '200' in black ink.

4 Clinical Particulars

4.9 Overdose

Clinical experience of overdose is limited. No overdoses of celecoxib were reported during clinical trials. Doses up to 2,400 mg/day for up to 10 days in 12 patients did not result in serious toxicity.
Signs and symptoms. Symptoms following acute NSAID overdoses are usually limited to lethargy, drowsiness, nausea, vomiting, epigastric pain and other gastrointestinal adverse effects, which are generally reversible with supportive care. Gastrointestinal bleeding can occur. Hypertension, acute renal failure, respiratory depression and coma may occur, but are rare.
Anaphylactoid reactions have been reported with therapeutic ingestion of NSAIDs, and may occur following an overdose.
Treatment of overdosage. There are no specific antidotes. Patients should be managed by symptomatic and supportive care following an overdose. Monitor patients for signs and symptoms of gastrointestinal ulceration and/or haemorrhage. Monitor serum electrolytes, renal function and urinalysis after significant overdose.
Consider activated charcoal in the event of a potentially toxic ingestion. Activated charcoal is most effective when administered within one or two hours of ingestion and may reduce absorption of the drug. In patients who are not fully conscious or have impaired gag reflex, consideration should be given to administering activated charcoal via a nasogastric tube, once the airway is protected.
No information is available regarding the removal of celecoxib by haemodialysis, but based on its high degree of plasma protein binding (> 97%) dialysis is unlikely to be useful in overdose. Forced diuresis, alkalinisation of urine, haemodialysis, or haemoperfusion may not be useful due to high protein binding.
For information on the management of overdose, contact the Poisons Information Centre on 13 11 26 (Australia).

5 Pharmacological Properties

5.3 Preclinical Safety Data

Genotoxicity. Celecoxib was not mutagenic in an Ames test and a mutation assay in Chinese hamster ovary (CHO) cells, nor clastogenic in a chromosome aberration assay in CHO cells and an in-vivo micronucleus test in rat bone marrow.
Carcinogenicity. Celecoxib was not carcinogenic in 2-year studies in rats given oral doses up to 200 mg/kg/day for males and 10 mg/kg/day for females (approximately 2-4 fold the human exposure as measured by the AUC0-24 h at 400 mg twice daily, which is twice the recommended maximum daily dose), or in mice given dietary doses up to 25 mg/kg/day for males and 50 mg/kg/day for females (slightly less than human exposure at 400 mg twice daily).

6 Pharmaceutical Particulars

6.7 Physicochemical Properties

Celecoxib is a diaryl substituted pyrazole.
Celecoxib is weakly acidic with a pKa in water of 11.1 and is practically insoluble in water, freely soluble to soluble in anhydrous ethanol and soluble in methylene chloride. Celecoxib is chemically unrelated to anti-inflammatory agents of steroidal or non-steroidal nature. Celecoxib does not contain a chiral centre.
Chemical structure.
https://stagingapi.mims.com/au/public/v2/images/fullchemgif/CSCELECO.gif Chemical name: 4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-yl] benzene sulfonamide.
Molecular formula: C17H14F3N3O2S.
Molecular weight: 381.37.
CAS number. 169590-42-5.

7 Medicine Schedule (Poisons Standard)

S4 - Prescription Only Medicine.

Summary Table of Changes

https://stagingapi.mims.com/au/public/v2/images/fulltablegif/CELBTCST.gif